TY - RPRT TI - Structural Characterization of Linker Shielding in ADC Site-Specific Conjugates AU - Jaime-Garza, Maru [Discovery Chemistry, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000336121739) AU - Waight, Andrew [Discovery Biologics, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000241101452) AU - Hudlikar, Manish [Discovery Chemistry, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000195232610) AU - Eddins, Michael J. [Discovery Chemistry, Merck & Co., Inc., 770 Sumneytown Pike, West Point, PA 19486, USA] (ORCID:0009000613711997) AU - Rasti, Elnaz S. [Discovery Biologics, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] AU - Zaragoza, Jan Paulo T. [Discovery Biologics, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000225836571) AU - Fayadat-Dilman, Laurence [Discovery Biologics, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000162858924) AU - Chrencik, Jill E. [Discovery Chemistry, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0009000563220478) AU - Gabelli, Sandra B. [Discovery Chemistry, Merck & Co., Inc., 770 Sumneytown Pike, West Point, PA 19486, USA] (ORCID:0000000312055204) AU - Chen, Yun-Ting [Discovery Chemistry, Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, USA] AU - Noland, Cameron L. [Discovery Chemistry, Merck & Co., Inc., 213 East Grand Ave., South San Francisco, CA 94080, USA] (ORCID:0000000163643167) PY - 2025 DO - 10.3390/pharmaceutics17121568 UR - https://www.osti.gov/biblio/3484928 ID - 3484928 ER -